Triazolopyrimidinedione

[1,2,4]Triazolo[1,5-a]pyrimidine-5,7(4H,6H)-dione





Reference:
Sci. Adv. 2021, 7, eabg4168.

Pyrimidinetrione

Pyrimidine-2,4,6(1H,3H,5H)-trione





Reference:
J. Med. Chem. 2025, 68, 21099-21119.

Cyclopropane

Reference:
Org. Lett. 2015, 17, 4944–4947.
The detailed experimental procedures can be found in the freely accessible Supporting Information.

Reference:
Org. Lett. 2015, 17, 4944–4947.
The detailed experimental procedures can be found in the freely accessible Supporting Information.

Triazole

Reference:
ACS Pharmacol. Transl. Sci. 2025, 8, 1072–1086.

Triazolopyrimidine

Triazolo[4,5-d]pyrimidine




Reference:
ACS Pharmacol. Transl. Sci. 2025, 8, 1072–1086.

Azauracil

Reference:
J. Med. Chem. 2014, 57, 3912-3923.
The detailed experimental procedures can be found in the freely accessible Supporting Information.

Pyridazinone

Pyridazin-4(1H)-one





Reference:
J. Med. Chem. 2014, 57, 22, 9627-9643.

Benzoimidazopyrimidine

1,4-Dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine

Reference:
J. Med. Chem. 2023, 66, 890-912.

Imidazopyridine

Imidazo[1,2-a]pyridine
Groebke–Blackburn–Bienaymé Multicomponent Reaction





Reference:
Monatsh Chem 2008, 139, 931-933.

4-Pyrone

Reference:
Org. Lett. 2007, 9, 2517-2520.